ATX inhibitor 1

ATX inhibitor 1是一种 ATX(IC50=1.23 nM, FS-3; 2.18 nM, bis-pNPP) 抑制剂。

CAS号

2225892-70-4

分子式

C21H23Cl2N2O6P

主要靶点

PDE

仅限科研使用

Cat No : CM05771

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Synonyms



产品信息

ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).

CAS号 2225892-70-4
分子式 C21H23Cl2N2O6P
主要靶点 PDE
主要通路 代谢
分子量 501.3
纯度 99.88%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 Powder: -20°C for 3 years | In solvent: -80°C for 1 year
别名

靶点活性

bis-pNPP:2.18 nM |FS-3:1.23 nM

溶解度

DMSO:250 mg/mL (498.70 mM),Sonification is recommended.

参考文献

1.Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409.

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