Carboxylesterase-IN-2

Carboxylesterase-IN-2 是一种有效的 Carboxylesterase Notum 抑制剂(IC50 ≤10 nM)。Carboxylesterase-IN-2具有研究癌症疾病的潜力。

CAS号

2764748-88-9

分子式

C13H12N4OS

主要靶点

Wnt/beta-catenin|Lipid

仅限科研使用

Cat No : CM14583

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Synonyms



产品信息

Carboxylesterase-IN-2 is a potent Carboxylesterase Notum inhibitor (IC50 ≤ 10 nM).Carboxylesterase-IN-2 has potential for the study of cancer diseases.

CAS号 2764748-88-9
分子式 C13H12N4OS
主要靶点 Wnt/beta-catenin|Lipid
主要通路 代谢|干细胞|细胞骨架
分子量 272.33
纯度 100.00%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件
别名

靶点活性

Carboxylesterase Notum:<10 nM

溶解度

DMSO:45.0 mg/mL (165.2 mM),Sonification is recommended.

参考文献

1.Steadman D, et al. Virtual Screening Directly Identifies New Fragment-Sized Inhibitors of Carboxylesterase Notum with Nanomolar Activity. J Med Chem. 2022;65(1):562-578.

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
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C1   V1   C2   V2