Nitrobenzylthioinosine

Nitrobenzylthioinosine (NBMPR) 是一种 ENT1 转运蛋白抑制剂,可与 ENT1 转运蛋白以高亲和力结合。它是一种可穿过血脑屏障的光亲和探针,用于追踪大脑中腺苷的摄取位点。

CAS号

38048-32-7

分子式

C17H17N5O6S

主要靶点

Adenosine Receptor|AChR

仅限科研使用

Cat No : CM03949

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Synonyms

NBMPR|S-(4-硝基苄基)-6-硫代肌苷



产品信息

Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.

CAS号 38048-32-7
分子式 C17H17N5O6S
主要靶点 Adenosine Receptor|AChR
主要通路 神经科学|G蛋白偶联受体
分子量 419.4
纯度 98.83%, 此纯度可做参考,具体纯度与批次有关系,可咨询客服
储存条件 Powder: -20°C for 3 years | In solvent: -80°C for 1 year
别名 NBMPR|S-(4-硝基苄基)-6-硫代肌苷

溶解度

DMSO:25 mg/mL (59.61 mM)

参考文献

1.P J Marangos, et al. [3H]nitrobenzylthioinosine is a photoaffinity probe for adenosine uptake sites in brain. Eur J Pharmacol. 1982 Dec 3;85(3-4):359-60.
2.C M Anderson, et al. Ability of nitrobenzylthioinosine to cross the blood-brain barrier in rats. Neurosci Lett. 1996 Nov 29;219(3):191-4.

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
×
=
×
C1   V1   C2   V2